Wholesale Small Molecules

Peptides & Small Molecules for Licensed Clinics

ExaVeyra Sciences supplies wholesale NAD+, glutathione, and bioactive small molecules to licensed clinics and practitioners nationwide. All formulations are organic chemist-verified, 503A/503B compliant, lyophilized for maximum stability, and backed by full COA documentation.

Organic Chemist-Verified503A/503B CompliantCOA on RequestLyophilizedThird-Party TestedLot TrackingNPI-Verified AccessIV/IM Ready

The Science

What Are Bioactive Small Molecules?

Bioactive small molecules are low-molecular-weight compounds that interact directly with biological systems at the cellular and subcellular level. Unlike large biologics such as proteins or antibodies, small molecules can cross cell membranes and engage intracellular targets — making them powerful tools for modulating cellular energy, redox balance, and metabolic function.

In regenerative and longevity medicine, small molecules like NAD+ precursors, coenzymes, and antioxidant tripeptides have emerged as foundational therapeutic agents. Their mechanisms are well-characterized in the biochemical literature, their safety profiles are established, and they integrate cleanly into IV therapy, functional medicine, and aesthetic protocols.

ExaVeyra's small molecule catalog is curated by our founder — an M.Sc. organic chemist — who evaluates every product against its underlying chemistry, manufacturing methodology, and analytical data. We supply only formulations that meet our documentation and purity standards, sourced through 503A/503B-compliant facilities.

Organic Chemist-Verified: Every small molecule in the ExaVeyra catalog is reviewed by our founder, Benn — an M.Sc. organic chemist with expertise in synthetic organic chemistry, analytical chemistry, and biochemistry. We go beyond COA review to evaluate the chemistry itself.

503A Compound Library

Every 503A Compound, One Searchable Library

Filter by therapeutic group or search by name, mechanism, or research area. Each compound has a dedicated page ready for peer-reviewed enrichment.

Showing 45 of 45 compounds

NAD+ (Nicotinamide Adenine Dinucleotide)

Nicotinamide Adenine Dinucleotide

Cellular Energy & DNA Repair
Format
Lyophilized (IV / IM)
Spec
250 mg, 500 mg
Group
Vitamins & IV Solutions

Research summary

Coenzyme in the mitochondrial electron transport chain and an obligate substrate for sirtuins (SIRT1-7) and PARP enzymes involved in DNA repair, genomic stability, and metabolic signaling.

View compound details2 citations

Compounded GLP-1 Formulation / B12

Compounded GLP-1 receptor agonist with Cyanocobalamin

GLP-1 Receptor Agonism
Format
Injectable
Spec
Multiple concentrations
Group
Weight Management

Research summary

GLP-1 receptor agonists activate incretin signaling to promote glucose-dependent insulin secretion, delay gastric emptying, and reduce appetite via central pathways.

View compound details1 citation

Compounded Dual-Incretin Formulation / B12

Compounded dual GIP / GLP-1 agonist with Cyanocobalamin

Dual Incretin Agonism
Format
Injectable
Spec
Multiple concentrations
Group
Weight Management

Research summary

Dual agonist acting on both GIP and GLP-1 receptors, enhancing glucose-dependent insulin release, improving lipid handling, and inducing greater weight reduction than GLP-1 monotherapy in clinical trials.

View compound details1 citation

Low Dose Naltrexone

Low Dose Naltrexone

Opioid Receptor Modulation
Format
Capsule
Spec
1.5 mg
Group
Hormone Optimization

Research summary

At sub-therapeutic doses, naltrexone transiently blocks opioid receptors, prompting compensatory upregulation of endogenous endorphin production and modulating microglial signaling.

View compound details1 citation

Glutathione

gamma-L-Glutamyl-L-cysteinylglycine

Master Antioxidant & Detoxification
Format
Injectable
Spec
200 mg/mL (10 mL, 30 mL)
Group
Vitamins & IV Solutions

Research summary

Endogenous tripeptide antioxidant. Primary substrate for glutathione peroxidase and glutathione S-transferase in phase II hepatic detoxification and reactive oxygen species neutralization.

View compound details1 citation

GHK-Cu 1%

Glycyl-L-histidyl-L-lysine copper(II) complex

Regenerative Copper Peptide
Format
Hair Restoration Solution
Spec
30 mL
Group
Hair Restoration

Research summary

Endogenous tripeptide-copper complex implicated in skin remodeling, angiogenesis, hair-follicle stimulation, and modulation of matrix metalloproteinases.

View compound details1 citation

Methylene Blue Anti-Aging Cream (0.0064% MB / 0.003% Estriol)

Methylthioninium chloride topical

Mitochondrial Electron Cycler
Format
Topical Cream
Spec
30 g
Group
Skin & Aesthetics

Research summary

Methylene blue cycles between oxidized and reduced forms, donating electrons to the mitochondrial electron transport chain and reducing reactive oxygen species in skin models.

View compound details1 citation

Compounded GLP-1 Formulation / Glycine

Compounded GLP-1 receptor agonist with Glycine

GLP-1 Receptor Agonism
Format
Injectable
Spec
Multiple concentrations
Group
Weight Management

Research summary

GLP-1 receptor agonist formulated with glycine as a stabilizing excipient in compounded preparations. Same mechanistic profile as semaglutide monotherapy.

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Compounded Dual-Incretin Formulation / Glycine

Compounded dual GIP / GLP-1 agonist with Glycine

Dual Incretin Agonism
Format
Injectable
Spec
Multiple concentrations
Group
Weight Management

Research summary

Glycine-buffered compounded dual-incretin formulation. Same receptor pharmacology as tirzepatide.

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DHEA

Dehydroepiandrosterone

Adrenal Hormone Precursor
Format
Capsule
Spec
25 mg / 50 mg / 100 mg
Group
Hormone Optimization

Research summary

Adrenal-derived C19 steroid precursor to both androgens and estrogens. Peripheral conversion is tissue-specific and declines with age.

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Branched Chain Amino Acids (BCAA: Isoleucine / Leucine / Valine)

Format
Injectable
Spec
30 mL
Group
Weight Management
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Glycine

Format
Injectable
Spec
50 mg/mL (10 mL)
Group
Weight Management
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Lipo-B (Cyanocobalamin / MIC)

Format
Injectable
Spec
10 mL, 30 mL
Group
Weight Management
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Lipo-C (Cyanocobalamin / MIC / L-Carnitine)

Format
Injectable
Spec
10 mL, 30 mL
Group
Weight Management
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Metformin HCl ER

Format
Tablet
Spec
500 mg and 1000 mg
Group
Weight Management
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Ondansetron (Zofran) 4 mg ODT

Format
Tablet
Spec
30 tablets (anti-nausea)
Group
Weight Management
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Bi-Est (80/20)

Format
Cream and Capsule
Spec
Multiple strengths
Group
Hormone Optimization
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Estradiol

Format
Capsule
Spec
0.25 mg–2 mg (multiple strengths)
Group
Hormone Optimization
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Estradiol

Format
Cream
Spec
Multiple strengths
Group
Hormone Optimization
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Progesterone

Format
Capsule (IR and SR)
Spec
Multiple strengths
Group
Hormone Optimization
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Progesterone

Format
Cream
Spec
Multiple strengths
Group
Hormone Optimization
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T4/T3 Combination

Format
Capsule (IR)
Spec
Multiple ratio strengths
Group
Hormone Optimization
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Liver Support (Vitamin E / Milk Thistle / NAC / Thiamine / Selenium)

Format
Capsule
Spec
Compounded formulation
Group
Hormone Optimization
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Ascorbic Acid (Vitamin C)

Format
Injectable
Spec
500 mg/mL (10 mL, 30 mL)
Group
Vitamins & IV Solutions
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Methylcobalamin (B12)

Format
Injectable
Spec
5 mg/mL (10 mL, 30 mL)
Group
Vitamins & IV Solutions
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Vitamin B-Complex (Thiamine / Niacinamide / Riboflavin-5-Phosphate / Pyridoxine)

Format
Injectable
Spec
30 mL
Group
Vitamins & IV Solutions
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Magnesium Chloride

Format
Injectable
Spec
200 mg/mL (50 mL)
Group
Vitamins & IV Solutions
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Biotin

Format
Injectable
Spec
10 mg/mL (10 mL)
Group
Vitamins & IV Solutions
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Vitamin D3

Format
Injectable
Spec
50,000 IU/mL (30 mL)
Group
Vitamins & IV Solutions
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Myers' Cocktail

Format
Injectable
Spec
10 mL, 30 mL
Group
Vitamins & IV Solutions
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Minoxidil 5% / Finasteride 0.1%

Format
Solution
Spec
60 mL
Group
Hair Restoration
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Minoxidil 5% / Tretinoin 0.025%

Format
Solution
Spec
60 mL
Group
Hair Restoration
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Minoxidil 5% / Azelaic Acid 12.5% / Finasteride 0.1% / Ketoconazole 2%

Format
Solution
Spec
60 mL
Group
Hair Restoration
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Finasteride

Format
Tablet
Spec
1 mg and 5 mg
Group
Hair Restoration
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Cashmere Cream (GHK-Cu 3% / Niacinamide 4%)

Format
Topical Cream
Spec
30 g
Group
Skin & Aesthetics
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GHK-Cu Biocosmetic Cream (GHK-Cu 3% / Estriol 0.003%)

Format
Topical Cream
Spec
30 g
Group
Skin & Aesthetics
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GHK-Cu Biocosmetic Cream + SNAP-8

Format
Topical Cream
Spec
30 g
Group
Skin & Aesthetics
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GHK-Cu 3% / SNAP-8 1% / Niacinamide 3% Serum

Format
Topical
Spec
30 mL
Group
Skin & Aesthetics
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GHK-Cu 3% / Niacinamide 3% Firm Boost Serum

Format
Topical
Spec
30 mL
Group
Skin & Aesthetics
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Ketoconazole 2% / Niacinamide 4%

Format
Cream
Spec
30 g
Group
Skin & Aesthetics
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Benzocaine 20% / Lidocaine 10% / Tetracaine 10%

Format
Topical Cream
Spec
60 mL pump
Group
Topical Numbing
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Lidocaine 23% / Tetracaine 10%

Format
Topical Cream
Spec
60 mL pump
Group
Topical Numbing
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Lidocaine 23% / Tetracaine 10% / Phenylephrine 0.5%

Format
Topical Cream
Spec
60 mL pump
Group
Topical Numbing
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Lidocaine 23% / Tetracaine 7% / Prilocaine 2%

Format
Topical Cream
Spec
60 mL pump
Group
Topical Numbing
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Phenylephrine

Format
Injectable
Spec
0.1%
Group
Topical Numbing
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Clinical Applications

How Clinics Use Our Small Molecules

Our practitioner network applies NAD+ and glutathione across a broad range of therapeutic and aesthetic specialties.

Longevity & Healthspan Research

NAD+ and supporting compounds for cellular energy restoration, mitochondrial optimization, and biological age management protocols.

IV Therapy & Infusion

Lyophilized formulations optimized for IV infusion and push protocols. Rapid reconstitution, clean purity profiles.

Detox & Antioxidant

Glutathione and antioxidant compounds for oxidative stress management, detoxification pathways, and immune support.

Aesthetic Medicine

Skin brightening, complexion optimization, and post-procedure recovery support using glutathione and regenerative compounds.

Functional Medicine

Metabolic support, mitochondrial health, and cellular repair protocols for functional and integrative medicine practices.

Surgical & Athletic Recovery

NAD+ and glutathione compounds used in post-surgical and post-training recovery protocols by licensed practitioners. Oxidative stress reduction and cellular energy metabolism are active areas of clinical research.

Quality & Compliance

503A/503B Compliant, Third-Party Tested

All ExaVeyra small molecule formulations are sourced through FDA-registered 503A and 503B compounding facilities. Every product undergoes third-party testing for purity, potency, and sterility. Certificates of analysis and lot tracking are available for every batch to support your practice's compliance requirements.

Lyophilized formulations are manufactured under strict aseptic conditions and tested for reconstitution performance. Our sourcing process is reviewed by an M.Sc. organic chemist who evaluates the underlying analytical methodology, including HPLC, mass spectrometry, and endotoxin testing, behind every product.

503A/503B Sourcing

Sourced exclusively through FDA-registered compounding facilities with documented quality systems.

Third-Party Tested

Independent purity, potency, and sterility testing on every lot. HPLC and mass spec verified.

Lyophilized Stability

Freeze-dried formulations with 2–3 year shelf life. No cold-chain required for storage.

Research summaries are provided for educational purposes. Connect with our compliance team before integrating any protocol.

Compliance & Research Team

Speak With Our Compliance Team

Our team can walk you through research context, sourcing questions, and regulatory considerations. Select any areas of interest and we'll connect you with the right specialist.

Areas of Interest Check all that apply

All inquiries are reviewed by our compliance and research team. We do not share your information with third parties.

Product Catalog

Small Molecule Products

NPI-verified wholesale pricing available after partner approval.

B1
Therapeutic Peptides in Orthopaedics: Applications, Challenges, and Future Directions
PMC Open Access · National Library of Medicine · 2025
View full publication ↗
B2
Injectable Therapeutic Peptides An Adjunct to Regenerative Medicine and Sports Performance?
Arthroscopy: The Journal of Arthroscopic and Related Surgery · Elsevier / Arthroscopy Association of North America · 2024
View full publication ↗
B3
Stable Gastric Pentadecapeptide BPC 157 and Wound Healing
Frontiers in Pharmacology · Frontiers Media · 2021
View full publication ↗
B4
Local and Systemic Peptide Therapies for Soft Tissue Regeneration: A Narrative Review
PMC Open Access · National Library of Medicine · 2024
View full publication ↗
⚠ EDUCATIONAL DISCLAIMER

The research citations and scientific content on this page are provided for educational and informational purposes only. This content does not constitute medical advice, diagnosis, or treatment recommendations. ExaVeyra Sciences does not make clinical efficacy claims for any products. All cited publications are independently authored peer-reviewed studies available through PubMed, PMC, or DOI. Practitioners should consult current FDA guidance and applicable regulations before clinical use.

Ready to Add NAD+ & Glutathione to Your Practice?

Apply for NPI-verified wholesale access to our full small molecule catalog. Team reviews applications within 1–3 business days.

Licensed healthcare providers only · NPI verification required · Miami-based, serving practices nationwide

Peptides & Small Molecules FAQ

How do medical practices order wholesale peptides?
Medical practices order wholesale peptides through verified B2B accounts that confirm professional credentials before pricing is shared. ExaVeyra Sciences supplies bioactive peptides with lot-specific certificates of analysis and HPLC purity documentation. Submit your NPI for verification, and our team will review current catalog availability and volume pricing tiers with your practice.
What purity standards apply to wholesale peptides for medical practices?
ExaVeyra's wholesale peptides are characterized by HPLC and mass spectrometry, with purity figures and identity confirmation reported on each certificate of analysis. Bioactive peptides are sourced from cGMP-aligned facilities and organic chemist-verified before release. Request a sample COA to review analytical standards before committing your practice to an order.
Are wholesale peptides for medical practices sourced compliantly?
ExaVeyra supplies bioactive peptides through 503A and 503B compliant sourcing channels and FDA-registered facilities, with documentation that supports your practice's recordkeeping. Practitioners apply peptides within their own scope and regulatory obligations. Our compliance team can review sourcing pathways and product status with your clinic before any purchase.
What formats are available when buying peptides wholesale?
ExaVeyra supplies wholesale peptides primarily in lyophilized form for stability, with documented storage parameters and reconstitution guidance. Each bioactive peptide ships with lot tracking and cold-chain handling where required. Contact our team to confirm available sequences, vial sizes, and volume pricing tiers matched to your practice.
How are wholesale peptides shipped and stored?
Wholesale peptides ship in temperature-controlled, lot-tracked packaging to preserve stability, and lyophilized bioactive peptides arrive with documented storage and reconstitution parameters. ExaVeyra includes a certificate of analysis with every shipment, so your practice has full analytical traceability. Ask our logistics team about delivery timelines in your state.

All compounded formulations are prepared by a licensed 503A sterile compounding pharmacy partner. Compounds are available to NPI-verified licensed practitioners only. Formulations are compounded per individual patient prescriptions in accordance with applicable state and federal law. Compounded medications are not FDA-approved. Pricing available upon verified account approval.

These statements have not been evaluated by the FDA. These products are not intended to diagnose, treat, cure, or prevent any disease. For licensed healthcare providers only. NPI verification required for wholesale access.