Opioid Receptor ModulationHormone Optimization503A Compounded

Low Dose Naltrexone

Low Dose Naltrexone

Format
Capsule
Spec
1.5 mg
Sourcing
FDA-registered 503A pharmacy

Research Summary

Mechanism & Physiological Role

At sub-therapeutic doses, naltrexone transiently blocks opioid receptors, prompting compensatory upregulation of endogenous endorphin production and modulating microglial signaling.

Clinical & Research Applications

Studied in the literature on autoimmune conditions, inflammatory pain, and fibromyalgia. Prescribing decisions are made by the treating practitioner.

Scientific Publications

Peer-Reviewed References

All compounded formulations are prepared by a licensed 503A sterile compounding pharmacy partner. Compounds are available to NPI-verified licensed practitioners only, per individual patient prescriptions in accordance with applicable state and federal law. Compounded medications are not FDA-approved. Pricing available upon verified account approval.

Ready to add Low Dose Naltrexone to your protocol?

Compounded formulations are dispensed by our licensed 503A pharmacy partner OBPRx under a valid patient-specific prescription. Prefer a formal quote? Request formulation-specific pricing instead.